LSD1/HDAC6-IN-1 是一种具有口服活性的组蛋白去甲基化酶 LSD1 和组蛋白去乙酰酶 HDAC6 (LSD1/HDAC6) 双重抑制剂，具有抗肿瘤活性。LSD1/HDAC6-IN-1 可用于多发性骨髓瘤 (MM) 的研究。
| 生物活性 | LSD1/HDAC6-IN-1 is an orally active dual inhibitor oflysine specific demethylase 1(LSD1)/Histone deacetylase 6 (HDAC6), with anti-tumor activity. LSD1/HDAC6-IN-1 can be used for the research of multiple myeloma (MM)[1]. |
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体外研究
(In Vitro) | LSD1/HDAC6-IN-1 shows superior potency in multiple MM lines[1].
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体内研究
(In Vivo) | LSD1/HDAC6-IN-1 is efficacy in the MM.1S xenograft model[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
