HDAC6-IN-9 (compound 12c) 是一种有效的选择性HDAC6抑制剂,HDAC1、HDAC3、HDAC6、HDAC8、HDAC10 的IC50值分别为 11.8, 15.2, 4.2, 139.6, 21.3 nM。HDAC6-IN-9 显示出抗增殖活性。
生物活性 | HDAC6-IN-9 (compound 12c) is a potent and selectiveHDAC6inhibitor withIC50values of 11.8, 15.2, 4.2, 139.6, 21.3 nM forHDAC1,HDAC3,HDAC6,HDAC8,HDAC10, respectively. HDAC6-IN-9 shows anti-proliferative activities[1]. |
IC50& Target[1] | HDAC1 11.8 nM (IC50) | HDAC3 15.2 nM (IC50) | HDAC6 4.2 nM (IC50) | HDAC8 139.6 nM (IC50) | HDAC10 21.3 nM (IC50) |
|
分子量 | |
Formula | |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |