(S)-HH2853 (compound 200) 是一种 PYRIDINO 五元芳环化合物,一种有效的EZH1/2双重抑制剂,对 EZH2_Y641F 的IC50为<100 nM。(S)-HH2853有潜力用于抗肿瘤或自身免疫性疾病的研究。
| 生物活性 | (S)-HH2853 (compound 200), a PYRIDINO five membered aromatic ring compound, is a potentEZH1/2dual inhibitor with anIC50of<100 nm for ezh2_y641f. (s)-hh2853 has the potential to be used in research of anti-tumor or autoimmune diseases[1]. |
| IC50& Target[1] | EZH1 | EZH2 Y641N <100 nM (IC50) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |