(R)-HH2853

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(R)-HH2853

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

2202678-06-4

(R)-HH2853 是一种突变型EZH2抑制剂，对EZH2-Y641F的IC₅₀<100 nM。(R)-HH2853 可用于癌症和自身免疫性疾病 (WO2018045971A1; compound 201)。

生物活性

(R)-HH2853 is amutantEZH2inhibitor with anIC₅₀of<100 nm forEZH2-Y641F. (R)-HH2853 can be used forcancerand autoimmune diseases (WO2018045971A1; compound 201)^[1].

IC₅₀& Target^[1]

EZH2 Y641F mutant type

<100 nM (IC₅₀)

分子量

611.66

Formula

C₃₁H₃₆F₃N₇O₃

CAS 号

2202678-06-4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.