CSV0C018875 是一种基于喹啉的EHMT2/G9a抑制剂。 CSV0C018875 的细胞毒性低于 BIX-01294。
| 生物活性 | CSV0C018875 is a quinoline-basedEHMT2/G9ainhibitor. CSV0C018875 exhibits lesser cytotoxicity than BIX-01294[1]. |
| IC50& Target[1] | |
体外研究
(In Vitro) | CSV0C018875 (2.5-20 μM; 48 hours) inhibits the levels of H3K9me2 modifications in the histones[1].
Western Blot Analysis[1] | Cell Line: | HEK293 cells | | Concentration: | 2.5 μM, 10 μM, 20 μM | | Incubation Time: | 48 hours | | Result: | Inhibited the enzymatic activity of G9a in a dose-dependent manner in HEK293 cells. |
|
| 分子量 | |
| Formula | |
| CAS 号 | |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
