Lintopride是5HT4拮抗剂,对5HT3 有轻微拮抗作用。
| 生物活性 | Lintopride is a5HT4antagonist with moderate 5HT3 antagonist properties. |
| IC50& Target[1] | 5-HT4Receptor | 5-HT3Receptor |
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体外研究 (In Vitro) | Lintopride significantly increases the lower oesophageal sphincter basal tone without affecting lower oesophageal sphincter physiological relaxation after swallowing. Peristaltic waves are also enhanced by Lintopride[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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