Sumatriptan (GR 43175 free base) 是一种具有口服活性的5-HT1受体激动剂，对5-HT1D、5-HT1B和5-HT1A受体的Ki分别为 17 nM、27 nM 和 100 nM。Sumatriptan 可用于偏头痛研究。
| 生物活性 | Sumatriptan (GR 43175 free base) is an orally active5-HT1 receptoragonist withKis of 17 nM, 27 nM and 100 nM for5-HT1D,5-HT1Band5-HT1A receptors, respectively. Sumatriptan can be used for migraine headache research[1][2]. |
| IC50& Target[1] | 5-HT1AReceptor 100 nM (Ki) | 5-HT1BReceptor 27 nM (Ki) | 5-HT1DReceptor 17 nM (Ki) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
