DR4485 hydrochloride

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本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

402942-53-4

DR4485 (hydrochloride) 是一种具有口服活性和选择性的 5-HT₇拮抗剂(pK_i=8.14)。

生物活性

DR4485 (hydrochloride) is an orally active and selective 5-HT₇antagonist (pK_i=8.14)^[1].

IC₅₀& Target^[1]

5-HT₇Receptor

8.14 (pKi)

体外研究
(In Vitro)

DR4485 (MZ54 WT cells; 6 μM or 8 μM) hydrochloride induces autophagy as well as cell death that is diminished by KO of ATG5 and ATG7^[2].

分子量

491.88

Formula

C₂₆H₂₉Cl₃N₂O

CAS 号

402942-53-4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.