3-Hydroxy agomelatine D3 是 3-Hydroxy agomelatine 的氘代物。3-Hydroxy agomelatine 是5-HT2C受体拮抗剂,IC50为 3.2 μM,Ki为 1.8 μM。
| 生物活性 | 3-Hydroxy agomelatine D3 is a deuterium labeled 3-Hydroxy agomelatine. 3-Hydroxy agomelatine is a5-HT2Creceptorantagonist with anIC50of 3.2 μM and aKiof 1.8 μM[1]. |
| IC50& Target[1] | 5-HT2CReceptor 3.2 μM (IC50) | 5-HT2CReceptor 1.8 μM (Ki) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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