LY-272015 hydrochloride 是一种具有口服活性的，特异性5-HT2B受体拮抗剂。LY-272015 hydrochloride 完全抑制 5-HT 或 BW723C86 诱导的 ERK2 磷酸化。LY-272015 hydrochloride 在醋酸去氧皮质酮 (DOCA)-盐高血压大鼠中具有抗高血压作用。
| 生物活性 | LY-272015 hydrochloride is an orally active, specific5-HT2Breceptorantagonist. LY-272015 hydrochloride completely inhibits the phosphorylation ofERK2induced by 5-HT or BW723C86. LY-272015 hydrochloride is antihypertensive in Deoxycorticosterone Acetate (DOCA)-salt-hypertensive rats[1][2]. |
| IC50& Target[1] | |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
