PSB 603 是一种有效且高度选择性的 A2B 腺苷受体拮抗剂，其 Ki 值为 0.553 nM，对人类和大鼠 A1 和 A2A 以及高达 10 μM 浓度的人类 A3 受体几乎没有亲和力。
| Cas No. | 1092351-10-4 |
| 化学名 | 8-(4-((4-(4-chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-2-hydroxy-1-propyl-1H-purin-6(7H)-one |
| Canonical SMILES | CCCN(C(O)=N1)C(C(N2)=C1N=C2C3=CC=C(S(N4CCN(C5=CC=C(Cl)C=C5)CC4)(=O)=O)C=C3)=O |
| 分子式 | C24H25ClN6O4S |
| 分子量 | 529.01 |
| 溶解度 | DMF: 5 mg/ml,DMSO: 5 mg/ml,DMSO:PBS(pH 7.2) (1:3): 0.25 mg/ml,Ethanol: slightly soluble |
| 储存条件 | Store at -20℃ |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
