CB1R antagonist 1

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CB1R antagonist 1

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

334668-69-8

CB1R Allosteric modulator 5 是一种选择性大麻素-1 受体 (CB1R) 逆向激动剂，其IC₅₀值为 4.2 μM 和EC₅₀值 >10 μM。CB1R Allosteric modulator 5 可用于代谢和肥胖的研究。

生物活性

CB1R Allosteric modulator 5, a selectivecannabinoid-1 receptor (CB1R)inverse agonist with anIC₅₀value of 4.2 μM andEC₅₀value of ＞10 μM. CB1R Allosteric modulator 5 can be used for the research of metabolic and obesity^[1].

IC₅₀& Target

hCB1-R

4.2 μM (IC₅₀)

hCB1-R

10 μM (EC₅₀)

体外研究
(In Vitro)

CB1R Allosteric modulator 5 has cannabinoid-1 receptor (CB1R) activity with an IC₅₀value of 4.2 μM and EC₅₀value of ＞10 μM^[1].

分子量

404.45

Formula

C₁₈H₂₃F₃N₂O₃S

CAS 号

334668-69-8

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.