(R)-Methanandamide (AM-356)，内源性大麻素配体 Anandamide 的类似物，是一种有效的CB1激动剂，Ki为 20 nM。(R)-Methanandamide 也能激活TRPV1受体。
| 生物活性 | (R)-Methanandamide (AM-356), an analog of the endocannabinoid ligand Anandamide, is a potentCB1agonist with aKiof 20 nM. (R)-Methanandamide also activatesvanilloid (TRPV1) receptors[1][2]. |
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体外研究
(In Vitro) | The endogenous cannabinoid (R)-Methanandamide exerts differential anti- and pronociceptive effects by activating both cannabinoid (CB1) and vanilloid (TRPV1) receptors of nociceptive primary afferents[2].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
