CB2R probe 1 是一种安全绿色的CB2R (2 型大麻素受体)荧光探针，Ki为 130 nM。CB2R probe 1 在癌细胞中显示出低细胞毒性。
| 生物活性 | CB2R probe 1 is a safe and greenCB2R (cannabinoid 2 receptor)fluorescent probe with anKiof 130 nM. CB2R probe 1 shows low cytotoxicity incancercells[1]. |
| IC50& Target[1] | cannabinoid type-2 receptors 130 nM (Ki) |
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体外研究
(In Vitro) | CB2R probe 1 (compound 28) (100 nM; 24 h) shows low cytotoxicity with IC50s of 1.6, 1.4, 1.4, 1.1, 2.6, 0.55, 2.0, 2.4, 2.8 nM for PANC1, U2OS, HT29, HT29-DX, U87AD, PC3, CB2R-HEK293, MCF7, MCFT-DX cells, respectively[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
