Antisauvagine-30 (aSvg-30) 是一种有效的、竞争性的、选择性的CRF2 receptor拮抗剂，针对小鼠 CRF2 细胞和大鼠 CRF1 受体的Kd值分别为 1.4 nM 和 153.6 nM。
| 生物活性 | Antisauvagine-30 (aSvg-30) is a potent, competitive and selectiveCRF2receptorantagonist withKdvalues of 1.4 nM and 153.6 nM for mouse CRF2β and rat CRF1 receptors, respectively[1]. |
| IC50& Target | Kd: 1.4 nM (mouse CRF2β);Kd: 153.6 nM (rat CRF1)[1] |
| 分子量 | |
| Formula | |
| CAS 号 | |
| Sequence | {D-Phe}-His-Leu-Leu-Arg-Lys-Met-Ile-Glu-Ile-Glu-Lys-Gln-Glu-Lys-Glu-Lys-Gln-Gln-Ala-Ala-Asn-Asn-Arg-Leu-Leu-Leu-Asp-Thr-Ile-NH2 |
| Sequence Shortening | (D-Phe)-HLLRKMIEIEKQEKEKQQAANNRLLLDTI-NH2 |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
