CXCR4 antagonist 3 (compound 12a) 是一种有效的CXCR4拮抗剂，IC50为 11 nM。CXCR4 antagonist 3 是 TIQ15 的同源物。CXCR4 antagonist 3 表现出最佳的整体特性，包括 CXCR4 拮抗、CYP 2D6 抑制、代谢稳定性和渗透性。CXCR4 antagonist 3 具有研究人类免疫缺陷病毒的潜力。
| 生物活性 | CXCR4 antagonist3 (compound 12a) is a potent antagonist ofCXCR4with anIC50of 11 nM.CXCR4 antagonist3 is a congener of TIQ15.CXCR4 antagonist3 demonstrates the best overall properties includingCXCR4antagonism, CYP 2D6 inhibition, metabolic stability, and permeability.CXCR4 antagonist3 has the potential for the research of human immunodeficiency virus[1]. |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
