COX-2-IN-28 是一种有效的选择性COX-2抑制剂,对COX-2, 15-LOX, COX-1 的IC50值分别为0.054, 2.14, 13.21μM。
| 生物活性 | COX-2-IN-28 is a potent and selectiveCOX-2inhibitor withIC50values of 0.054, 2.14, 13.21 μM forCOX-2,15-LOX,COX-1,respectively[1]. |
| IC50& Target[1] | COX-1 13.21 μM (IC50) | COX-2 0.054 μM (IC50) | 15-LOX 2.14 μM (IC50) |
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体外研究 (In Vitro) | COX-2-IN-28 (compound 15c) shows significant COX-2 selectivity with an SI value of 244.63[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |