Alimemazine 是通常用作止痒剂的吩噻嗪衍生物,也是血凝素 (HA)- 受体的拮抗剂。Alimemazine (Trimeprazine) 是也是针对组胺H1受体 (H1R) 和其他 GPCR 的部分激动剂。Alimemazine 具有抗血清素、抗痉挛和止吐作用。
生物活性 | Alimemazine is a phenothiazine derivative that is generally used as an antipruritic agent and also ahemagglutinin(HA)-receptorantagonist.Alimemazine (Trimeprazine) is also acts as a partial agonist against the histamine H1 receptor (H1R) and other GPCRs. Alimemazine displays antiserotonin, antispasmodic, and antiemetic properties[1][2]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |