Doxepin D3 Hydrochloride 是 Doxepin Hydrochloride 的氘代物。Doxepin hydrochloride 是一种口服活性的三环抗抑郁药。Doxepin hydrochloride 是一种有效的选择性组胺受体H1拮抗剂。Doxepin hydrochloride 也是一种有效的CYP450抑制剂,并显着抑制CYP450 2C19和CYP450 1A2。
| 生物活性 | Doxepin D3 Hydrochloride is a deuterium labeled Doxepin Hydrochloride. Doxepin hydrochloride is an orally active tricyclic antidepressant. Doxepin hydrochloride is a potent and selectivehistamine receptorH1antagonist. Doxepin hydrochloride is also a potentCYP450inhibitor and significantly inhibitsCYP450 2C19and1A2[1][2]. |
| IC50& Target | Histamine receptor H1; CYP450 2C19 and CYP450 1A2[2] |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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