EGFR/ErbB-2/ErbB-4 inhibitor-3 (compound 29) 是一种有效的酪氨酸激酶抑制剂,erbB1、erbB2、erbB4、EGF、HER 的IC50s 分别为 0.3、 1.1、0.5、2.5、24 nM。
| 生物活性 | EGFR/ErbB-2/ErbB-4 inhibitor-3 (compound 29) is a potenttyrosine kinaseinhibitor withIC50s of 0.3, 1.1, 0.5, 2.5, 24 nM for erbB1, erbB2, erbB4,EGF, HER, respectively[1]. |
| IC50& Target[1] | ErbB2 1.1 nM (IC50) | ErbB1 0.3 nM (IC50) | ErbB4 0.5 nM (IC50) | EGFR 2.5 nM (IC50) | HER 24 nM (IC50) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |