ERK2 IN-1 是一种选择性ERK2抑制剂，IC50为 7 nM。
| 生物活性 | ERK2IN-1 is a selectiveERK2inhibitor with anIC50of 7 nM[1]. |
| IC50& Target[1] | |
体外研究
(In Vitro) | ERK1/2 IN-1 (Compound 28) maintains good ERK enzymatic activity (ERK IC50=7 nM) and cellular activity in BRAF/KRAS mutant wildtype cancer cell lines (HT-29/Caspase IC50=118/80 nM)[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
