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(R)-Baclofen hydrochloride
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
(R)-Baclofen hydrochloride图片
CAS NO:63701-55-3

(R)-巴氯芬盐酸盐
Arbaclofen hydrochloride
STX 209 hydrochloride
(R)-Baclofen hydrochloride (Arbaclofen hydrochloride) 是选择性GABAB受体激动剂。
生物活性

(R)-Baclofen hydrochloride (Arbaclofen hydrochloride) is a selectiveGABAB receptoragonist[1][2].

IC50& Target

GABAB receptor[1]

体内研究
(In Vivo)

(R)-Baclofen hydrochloride (STX 209 hydrochloride) suppresses audiogenic seizures in theFmr1-knockout mouse on the seizure-resistant C57BL/6 background with an effective dose of 1 mg/kg[3].
Acute intraperitoneal administration of (R)-Baclofen hydrochloride significantly reduces the percent of mice displaying seizures (seizure incidence), with a minimum effective dose (MED) of 1.5 mg/kg[3].

Clinical Trial
分子量

250.12

Formula

C10H13Cl2NO2

CAS 号

63701-55-3

中文名称

(R)-巴氯芬盐酸盐;(R)-氯苯氨丁酸盐酸盐

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

 
 
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