Tilapertin 是甘氨酸转运蛋白 1 型 (GlyT1) 的口服抑制剂。
| 生物活性 | Tilapertin is an oral inhibitor of glycine transporter type-1 (GlyT1). |
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体内研究
(In Vivo) | Tilapertin is a nanomolar potent, orally bioavailable and selective GlyT1 inhibitor. Oral administration of Tilapertin dose-dependently increases cerebrospinal fluid (CSF) glycine concentration in rats[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
