PSB 36 是一种有效的选择性腺苷 A1 受体拮抗剂,对 rA1、hA2B、rA2A、hA3 和 rA3 受体的 Kis 值分别为 0.12 nM、187 nM、552 nM、2300 nM 和 6500 nM。
Cas No. | 524944-72-7 |
化学名 | 1-butyl-3-(3-hydroxypropyl)-8-((2R,3as,5S,6ar)-octahydro-2,5-methanopentalen-3a-yl)-1H-purine-2,6(3H,7H)-dione |
Canonical SMILES | O=C1N(CCCC)C(N(CCCO)C2=C1NC([C@@]3(C[C@H]4C5)[C@@H]5C[C@H](C4)C3)=N2)=O |
分子式 | C21H30N4O3 |
分子量 | 386.49 |
溶解度 | <38.65mg/ml in ethanol;<38.65mg/ml in DMSO |
储存条件 | Store at -20℃ |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |